Kenneth J. Linton

Repacking of the transmembrane domains of P-glycoprotein during the transport ATPase cycle

Rosenberg, Mark F., Velarde, Giles, Ford, Robert C., Martin, Catherine, Berridge, Georgina, Kerr, Ian D., ...

P-glycoprotein (P-gp) is an ABC (ATP-binding cassette) transporter, which hydrolyses ATP and extrudes cytotoxic drugs from mammalian cells. P-gp consists of two transmembrane domains (TMDs) that span...

Repacking of the transmembrane domains of P-glycoprotein during the transport ATPase cycle

Rosenberg, Mark F., Velarde, Giles, Ford, Robert C., Martin, Catherine, Berridge, Georgina, Kerr, Ian D., ...

P-glycoprotein (P-gp) is an ABC (ATP-binding cassette) transporter, which hydrolyses ATP and extrudes cytotoxic drugs from mammalian cells. P-gp consists of two transmembrane domains (TMDs) that span...

Detailed characterization of cysteine-less P-glycoprotein reveals subtle pharmacological differences in function from wild-type protein

Taylor, Andrew M, Storm, Janet, Soceneantu, Loredana, Linton, Kenneth J, Gabriel, Mark, Martin, Catherine, ...

Subtle alterations in the coupling of drug binding to nucleotide hydrolysis were observed following mutation of all seven endogenous cysteine residues to serines in the human multidrug resistance...

Cd36, a class B scavenger receptor, functions as a monomer to bind acetylated and oxidized low-density lipoproteins

Martin, Catherine A., Longman, Emma, Wooding, Carol, Hoosdally, Sarah J., Ali, Saira, Aitman, Timothy J., ...

Cd36 is a small-molecular-weight integral membrane protein expressed in a diverse, but select, range of cell types. It has an equally diverse range of ligands and physiological functions, which has...